Emoxypine Succinate powder
Emoxypine Succinate powder

Emoxypine Succinate powder

Product Code: CAS:27464-43-1
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Product Summary:

Emoxypine (a.k.a. Mexidol, Mexifin - specifically within its succinate salt form), is an unusually pleiotropic anti-oxidant with structural resemblance to pyridoxine with several research indications.  Indications include anxiolytic, nootropic, neuroprotective, antidepressant, anti-hypoxic, and anti-addictive research.

Product Description

Synonyms:mexidol

Formal Name:MODAFINIL-DEA SCHEDULE IV;CRL-40476

Formula   C8H11NO.C4H6O4

Molecular Weight: 273.35 g/mol

Purity≥99%

CAS Number: 127464-43-1

Other names

mexidol;2-Ethyl-6-methyl-3-pyridinol butanoate (1:1);2-Ethyl-6-methyl-3-hydroxypyridine succinate;Butanedioic acid 2-ethyl-6-methyl-3-pyridinol (1:1);2-Ethyl-6-Methylpyridin-3-ol succinate;2-ethyl-6-Methyl-3-hydroxypyridine succinate (Mexidole);2-Ethyl-6-Methyl-3-pyridinol butanoate;Mexidole (2-ethyl-6-Methyl-3-hydroxypyridine succinate)

What Is Emoxypine Succinate?

Emoxypine was first synthesized by L.D. Smirnov and K.M. Dumayev, then studied and developed in the Institute of Pharmacology, Russian Academy of Medical Sciences and National Scientific Center of Bioactive Substances Safety.

History of Emoxypine Succinate

Emoxypine was first synthesized by L.D. Smirnov and K.M. Dumayev, then studied and developed in the Institute of Pharmacology, Russian Academy of Medical Sciences and National Scientific Center of Bioactive Substances Safety.

Emoxypine Succinate USES

In Russia, emoxypine has a wide range of applications in medical practice. It purportedly exercises anxiolytic, anti-stress, anti-alcohol, anticonvulsant, nootropic, neuroprotective and anti-inflammatory action.Emoxypine presumably improves cerebral blood circulation, inhibits thrombocyte aggregation, lowers cholesterol levels, has cardioprotective and antiatherosclerotic action.

Emoxypine Succinate Chemical Structure

Formula   C8H11NO

Molecular mass:137.179 g/mol

SMILES:CCc1c(ccc(n1)C)O

InChI

InChI=1S/C8H11NO/c1-3-7-8(10)5-4-6(2)9-7/h4-5,10H,3H2,1-2H3

Key:JPGDYIGSCHWQCC-UHFFFAOYSA-N

Melting point:170 to 172 °C (338 to 342 °F)

Emoxypine Succinate Mechanism of Action

Emoxypine's mechanism of action is believed to be its antioxidant and membrane-protective effects with the following key components:

Emoxypine effectively inhibits free radical oxidation of biomembrane lipids, reacts to peroxide radicals of lipids primary and hydroxyl radical of peptides Increases the activity of antioxidant enzymes, specifically that of superoxide dismutase, responsible for the formation and consumption of lipid peroxides and active oxygen forms Inhibits free radicals during the synthesis of prostaglandin catalyzed cyclooxygenase and lipoxygenase, increases the correlation prostacyclin/ thromboxane A2 and blocks the leukotriene formation Increases the content of polar fraction of lipids (phosphatidyl serine and phosphatidyl inositol) and reduces the cholesterol/phospholipids ratio which proves its lipid-regulatory properties; shifts structure transition into the low temperature zones, that is provokes the reduction of membrane viscosity and the increase of its fluidity, increases lipid-protein ration.

Modulates the activity of membrane-bound enzymes: phosphodiesterase, cyclic nucleotides, adenylate cyclase, aldoreductase, acetylcholinesterase.

Modulates the receptor complexes of the brain membranes, i.e. benzodiazepine, GABA, acetylcholine receptors by increasing their binding ability.

Stabilizes biomembranes, i.e. membrane structures of blood cells - erythrocytes and thrombocytes during their haemolysis or mechanical injury accompanied by the formation of free radicals.

Changes the monoamine level and increases the dopamine content in the brain.

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